SCHEMBL20121610

SCHEMBL20121610

O=C(CCc1ccc(F)cc1)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(F)cc2)C1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.70
CYP3A4 P08684 1/20 0.49
MLNR O43193 1/20 0.42
ME2 P23368 1/20 0.41
ME1 P48163 1/20 0.41
ME3 Q16798 1/20 0.41
GFER P55789 1/20 0.41
CACNA1F O60840 1/20 0.39
HTR1A P08908 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
DRD4 P21917 1/20 0.39
DRD5 P21918 1/20 0.39
HRH2 P25021 1/20 0.39
ADRA1D P25100 1/20 0.39
HTR2A P28223 1/20 0.39
HTR7 P34969 1/20 0.39
ADRA1A P35348 1/20 0.39
HRH1 P35367 1/20 0.39
ADRA1B P35368 1/20 0.39
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17636399 0.95 KCNH2 (0.78) KCNH2CYP3A4MLNRME2ME1
SCHEMBL20121576 0.95 KCNH2 (0.78) KCNH2CYP3A4MLNRME2ME1
SCHEMBL20121554 0.95 KCNH2 (0.68) KCNH2CYP3A4MLNRME2ME1
SCHEMBL20121613 0.95 KCNH2 (0.78) KCNH2CYP3A4MLNRME2ME1
SCHEMBL12951885 0.95 KCNH2 (0.67) KCNH2CYP3A4GFER
SCHEMBL20121599 0.93 KCNH2 (0.68) KCNH2CYP3A4MLNRME2ME1
SCHEMBL20121570 0.93 KCNH2 (0.64) KCNH2CYP3A4MLNR
SCHEMBL12952261 0.92 KCNH2 (0.73) KCNH2CYP3A4MLNRME2ME1
SCHEMBL12952248 0.91 KCNH2 (0.75) KCNH2CYP3A4MLNR
SCHEMBL15760176 0.91 KCNH2 (0.72) KCNH2CYP3A4MLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed