SCHEMBL20121561

SCHEMBL20121561

CC(C)(C)CC(=O)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(Cl)cc2)C1

nearest known ligand 0.76

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.76
CYP3A4 P08684 1/20 0.48
P2RX7 Q99572 2/20 0.41
SLC2A1 P11166 1/20 0.41
CSNK1D P48730 1/20 0.40
CSNK1E P49674 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
TGFBR1 P36897 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12952046 0.95 KCNH2 (0.74) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL20121586 0.92 KCNH2 (0.80) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL12952195 0.90 KCNH2 (0.74) KCNH2CYP3A4P2RX7PTGDR2
SCHEMBL20121558 0.90 KCNH2 (0.80) KCNH2CYP3A4P2RX7CSNK1DCSNK1E
SCHEMBL2069248 0.88 KCNH2 (0.71) KCNH2CYP3A4P2RX7CSNK1DCSNK1E
SCHEMBL1052384 0.88 KCNH2 (0.82) KCNH2CYP3A4P2RX7PTGDR2TGFBR1
SCHEMBL2067454 0.88 KCNH2 (0.82) KCNH2CYP3A4P2RX7PTGDR2TGFBR1
SCHEMBL12952051 0.87 KCNH2 (0.70) KCNH2CYP3A4P2RX7PTGDR2
SCHEMBL12952054 0.87 KCNH2 (0.70) KCNH2CYP3A4P2RX7SLC2A1PTGDR2
SCHEMBL2068537 0.86 KCNH2 (1.00) KCNH2CYP3A4P2RX7CSNK1DCSNK1E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed