SCHEMBL20121586

SCHEMBL20121586

Cc1ccc(Nc2c(-c3ccc(F)cc3)nc3n2CCN(C(=O)CC(C)(C)C)C3)cc1

nearest known ligand 0.80

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.80
CYP3A4 P08684 1/20 0.49
CSNK1D P48730 1/20 0.39
CSNK1E P49674 1/20 0.39
TGFBR1 P36897 2/20 0.38
TP53 P04637 2/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
DPP4 P27487 1/20 0.36
DPP8 Q6V1X1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12952046 0.96 KCNH2 (0.74) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL2068457 0.94 KCNH2 (0.78) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL2070871 0.92 KCNH2 (0.76) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL20121561 0.92 KCNH2 (0.76) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL2069762 0.91 KCNH2 (0.75) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL1051468 0.89 KCNH2 (0.77) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL15760130 0.89 KCNH2 (0.71) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL1050387 0.89 KCNH2 (0.82) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL1048701 0.89 KCNH2 (1.00) KCNH2CYP3A4TGFBR1TP53MAPT
SCHEMBL998631 0.89 KCNH2 (1.00) KCNH2CYP3A4TGFBR1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed