SCHEMBL20121565

SCHEMBL20121565

Cc1ccc(Nc2c(-c3ccc(F)c(F)c3)nc3n2CCN(C(=O)CCc2ccc(F)c(F)c2)C3)cc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.63
DPP4 P27487 3/20 0.38
DPP8 Q6V1X1 3/20 0.38
DPP7 Q9UHL4 2/20 0.38
CYP3A4 P08684 1/20 0.38
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
P2RX7 Q99572 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20121557 0.95 KCNH2 (0.71) KCNH2DPP4DPP8DPP7CYP3A4
SCHEMBL20121570 0.91 KCNH2 (0.64) KCNH2DPP4DPP8DPP7CYP3A4
SCHEMBL2067372 0.91 KCNH2 (0.66) KCNH2DPP4DPP8DPP7CYP3A4
SCHEMBL15760180 0.90 KCNH2 (0.69) KCNH2DPP4DPP8CYP3A4ALDH1A1
SCHEMBL12952184 0.89 KCNH2 (0.68) KCNH2DPP4DPP8DPP7CYP3A4
SCHEMBL20121595 0.88 KCNH2 (0.67) KCNH2DPP4DPP8DPP7CYP3A4
SCHEMBL17636399 0.88 KCNH2 (0.78) KCNH2CYP3A4ALDH1A1KMT2AMEN1
SCHEMBL20121576 0.88 KCNH2 (0.78) KCNH2CYP3A4ALDH1A1KMT2AMEN1
SCHEMBL998387 0.88 KCNH2 (0.81) KCNH2DPP4DPP8DPP7CYP3A4
SCHEMBL20121613 0.88 KCNH2 (0.78) KCNH2CYP3A4ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed