SCHEMBL20121576

SCHEMBL20121576

Cc1ccc(CCC(=O)N2CCn3c(nc(-c4ccc(F)cc4)c3Nc3ccc(F)cc3)C2)cc1

nearest known ligand 0.78

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.78
CYP3A4 P08684 1/20 0.48
MLNR O43193 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
MAPK1 P28482 1/20 0.39
ME2 P23368 1/20 0.39
ME1 P48163 1/20 0.39
ME3 Q16798 1/20 0.39
GPBAR1 Q8TDU6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20121613 1.00 KCNH2 (0.78) KCNH2CYP3A4MLNRALDH1A1KMT2A
SCHEMBL17636399 1.00 KCNH2 (0.78) KCNH2CYP3A4MLNRALDH1A1KMT2A
SCHEMBL12952261 0.97 KCNH2 (0.73) KCNH2CYP3A4MLNRALDH1A1KMT2A
SCHEMBL20121603 0.96 KCNH2 (0.78) KCNH2CYP3A4MLNRALDH1A1KMT2A
SCHEMBL20121572 0.96 KCNH2 (0.72) KCNH2CYP3A4MLNRALDH1A1KMT2A
SCHEMBL15760176 0.96 KCNH2 (0.72) KCNH2CYP3A4MLNRALDH1A1KMT2A
SCHEMBL12952248 0.96 KCNH2 (0.75) KCNH2CYP3A4MLNRALDH1A1KMT2A
SCHEMBL12952250 0.96 KCNH2 (0.75) KCNH2CYP3A4
SCHEMBL20121610 0.95 KCNH2 (0.70) KCNH2CYP3A4MLNRME2ME1
SCHEMBL12952166 0.95 KCNH2 (0.71) KCNH2CYP3A4MLNRALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed