SCHEMBL20121580

SCHEMBL20121580

Cc1ccc(Nc2c(-c3ccc(F)c(F)c3)nc3n2CCN(C(=O)CC(C)C)C3)cc1

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.65
TACR3 P29371 1/20 0.40
DPP4 P27487 5/20 0.40
DPP8 Q6V1X1 5/20 0.40
DPP7 Q9UHL4 2/20 0.39
CYP3A4 P08684 1/20 0.39
ATM Q13315 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MDM2 Q00987 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12952184 0.90 KCNH2 (0.68) KCNH2TACR3DPP4DPP8DPP7
SCHEMBL12782067 0.90 KCNH2 (0.80) KCNH2TACR3DPP4DPP8CYP3A4
SCHEMBL998387 0.89 KCNH2 (0.81) KCNH2DPP4DPP8DPP7CYP3A4
SCHEMBL12952188 0.89 KCNH2 (0.71) KCNH2TACR3DPP4DPP8DPP7
SCHEMBL2067372 0.89 KCNH2 (0.66) KCNH2DPP4DPP8DPP7CYP3A4
SCHEMBL2068398 0.87 KCNH2 (0.61) KCNH2DPP4DPP8CYP3A4
SCHEMBL20121565 0.86 KCNH2 (0.63) KCNH2DPP4DPP8DPP7CYP3A4
SCHEMBL12952270 0.86 KCNH2 (0.73) KCNH2TACR3DPP4DPP8CYP3A4
SCHEMBL2068807 0.86 KCNH2 (0.58) KCNH2TACR3CYP3A4
SCHEMBL2068091 0.85 KCNH2 (0.59) KCNH2DPP4DPP8DPP7CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed