SCHEMBL20121585

SCHEMBL20121585

CC1=NC(=O)Cn2c1nc(-c1ccc(F)cc1)c2Nc1ccc(Cl)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.54
CYP3A4 P08684 1/20 0.37
RAPGEF4 Q8WZA2 1/20 0.36
AXL P30530 1/20 0.36
MAPT P10636 2/20 0.35
POLB P06746 1/20 0.35
KCNK3 O14649 1/20 0.35
GSK3B P49841 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20121571 0.89 KCNH2 (0.51) KCNH2CYP3A4RAPGEF4AXLKCNK3
SCHEMBL20121615 0.88 KCNH2 (0.52) KCNH2CYP3A4MAPT
SCHEMBL20121614 0.76 KCNH2 (0.49) KCNH2CYP3A4MAPT
SCHEMBL1050256 0.76 KCNH2 (0.52) KCNH2CYP3A4RAPGEF4AXLMAPT
SCHEMBL1048591 0.76 KCNH2 (0.54) KCNH2CYP3A4AXLMAPTKDM4E
SCHEMBL1050163 0.76 KCNH2 (0.52) KCNH2CYP3A4RAPGEF4AXLMAPT
SCHEMBL1051207 0.74 KCNH2 (0.50) KCNH2CYP3A4AXLMAPTPOLB
SCHEMBL20121581 0.74 KCNH2 (0.50) KCNH2CYP3A4AXLMAPTPOLB
SCHEMBL1051425 0.74 KCNH2 (0.50) KCNH2CYP3A4AXLMAPTPOLB
SCHEMBL2068748 0.73 KCNH2 (0.62) KCNH2CYP3A4MEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed