SCHEMBL20121615

SCHEMBL20121615

CC1=NC(=O)Cn2c1nc(-c1ccc(F)cc1)c2Nc1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.52
CYP3A4 P08684 1/20 0.41
MAPT P10636 5/20 0.40
GAA P10253 4/20 0.40
TP53 P04637 3/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TUBB4A P04350 2/20 0.36
TUBB P07437 2/20 0.36
TUBA3C P0DPH7 2/20 0.36
TUBA1B P68363 2/20 0.36
TUBA4A P68366 2/20 0.36
TUBB4B P68371 2/20 0.36
TUBB3 Q13509 2/20 0.36
TUBB2A Q13885 2/20 0.36
TUBB8 Q3ZCM7 2/20 0.36
TUBA3E Q6PEY2 2/20 0.36
TUBA1A Q71U36 2/20 0.36
TUBA1C Q9BQE3 2/20 0.36
TUBB6 Q9BUF5 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20121585 0.88 KCNH2 (0.54) KCNH2CYP3A4MAPT
SCHEMBL20121614 0.88 KCNH2 (0.49) KCNH2CYP3A4MAPTGAATP53
SCHEMBL20121571 0.76 KCNH2 (0.51) KCNH2CYP3A4
SCHEMBL1050451 0.74 KCNH2 (0.60) KCNH2CYP3A4MAPTGAATP53
SCHEMBL1049863 0.74 KCNH2 (0.49) KCNH2CYP3A4MAPTGAATP53
SCHEMBL1052381 0.74 KCNH2 (0.49) KCNH2CYP3A4MAPTGAATP53
SCHEMBL2068872 0.72 KCNH2 (0.47) KCNH2CYP3A4MAPTGAATP53
SCHEMBL1050385 0.71 KCNH2 (0.55) KCNH2CYP3A4MAPTGAATP53
SCHEMBL2068857 0.70 KCNH2 (0.68) KCNH2CYP3A4MAPTGAATP53
SCHEMBL12952195 0.69 KCNH2 (0.74) KCNH2CYP3A4MAPTPTGDR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed