SCHEMBL20121592

SCHEMBL20121592

CCC(=O)Nc1ccc(CCC(=O)N2CCn3c(nc(-c4cccc(F)c4)c3Nc3ccc(F)cc3)C2)cc1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 11/20 0.62
POLB P06746 1/20 0.46
MLNR O43193 2/20 0.39
CSNK1D P48730 1/20 0.39
CSNK1E P49674 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.38
MCHR1 Q99705 1/20 0.37
MAPK10 P53779 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20121591 0.93 KCNH2 (0.60) KCNH2POLBMLNRCSNK1DCSNK1E
SCHEMBL20121604 0.91 KCNH2 (0.59) KCNH2POLBMLNRCSNK1DCSNK1E
SCHEMBL12952023 0.89 KCNH2 (0.69) KCNH2POLBMLNRCYP3A4MCHR1
SCHEMBL997790 0.86 KCNH2 (0.62) KCNH2CSNK1DCSNK1ECYP3A4
SCHEMBL20121541 0.85 KCNH2 (0.57) KCNH2POLBMLNRCSNK1EMAPT
SCHEMBL20121610 0.84 KCNH2 (0.70) KCNH2MLNRCYP3A4MCHR1
SCHEMBL12952035 0.84 KCNH2 (0.66) KCNH2CSNK1DCSNK1ECYP3A4MAPT
SCHEMBL12952031 0.84 KCNH2 (0.68) KCNH2POLBMLNRCYP3A4MAPT
SCHEMBL12951892 0.83 KCNH2 (0.56) KCNH2CSNK1DCSNK1ECYP3A4MAPT
SCHEMBL20121567 0.82 KCNH2 (0.63) KCNH2CSNK1DCSNK1ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed