SCHEMBL20121600

SCHEMBL20121600

CCCNC(=O)CCC(=O)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(C)cc2)C1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.73
CYP3A4 P08684 1/20 0.45
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
TP53 P04637 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
TGFBR1 P36897 2/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20121553 0.95 KCNH2 (0.71) KCNH2CYP3A4MEN1KMT2ATP53
SCHEMBL12952259 0.90 KCNH2 (0.69) KCNH2CYP3A4MEN1KMT2ATP53
SCHEMBL12952026 0.90 KCNH2 (0.78) KCNH2CYP3A4MEN1KMT2ATGFBR1
SCHEMBL12952020 0.89 KCNH2 (0.77) KCNH2CYP3A4MEN1KMT2ATGFBR1
SCHEMBL12952035 0.88 KCNH2 (0.66) KCNH2CYP3A4TAAR1
SCHEMBL1051800 0.88 KCNH2 (0.76) KCNH2CYP3A4TGFBR1
SCHEMBL2069249 0.88 KCNH2 (0.81) KCNH2CYP3A4TP53TGFBR1
SCHEMBL1046563 0.87 KCNH2 (0.65) KCNH2CYP3A4MEN1KMT2ATP53
SCHEMBL1051024 0.86 KCNH2 (0.66) KCNH2CYP3A4MEN1KMT2ATP53
SCHEMBL20121576 0.86 KCNH2 (0.78) KCNH2CYP3A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed