SCHEMBL20123280

SCHEMBL20123280

C/C(=C/C1=C(Cl)C(=N)c2ccccc2C1=O)C(=O)O

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 14/20 0.78
AKR1C3 P42330 1/20 0.44
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
S100A4 P26447 1/20 0.40
IDO1 P14902 1/20 0.38
DNMT1 P26358 1/20 0.38
DNMT3L Q9UJW3 1/20 0.38
DNMT3A Q9Y6K1 1/20 0.38
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
APAF1 O14727 1/20 0.36
TDP2 O95551 1/20 0.36
NSD2 O96028 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3743465 0.88 APEX1 (1.00) APEX1AKR1C3HSP90AA1HSP90AB1IDO1
SCHEMBL3745788 0.88 APEX1 (1.00) APEX1AKR1C3HSP90AA1HSP90AB1IDO1
SCHEMBL3743461 0.88 APEX1 (1.00) APEX1AKR1C3HSP90AA1HSP90AB1IDO1
SCHEMBL20123229 0.85 APEX1 (0.57) APEX1HSP90AA1HSP90AB1S100A4KDM4E
SCHEMBL13894618 0.83 APEX1 (0.78) APEX1AKR1C3HSP90AA1HSP90AB1IDO1
SCHEMBL13894584 0.83 APEX1 (0.78) APEX1AKR1C3HSP90AA1HSP90AB1IDO1
SCHEMBL3745792 0.80 APEX1 (1.00) APEX1AKR1C3S100A4KDM4EAPAF1
SCHEMBL3745796 0.80 APEX1 (1.00) APEX1AKR1C3S100A4KDM4EAPAF1
SCHEMBL20123275 0.80 APEX1 (0.82) APEX1HSP90AA1HSP90AB1KDM4EMAPT
SCHEMBL3748323 0.77 APEX1 (1.00) APEX1AKR1C3HSP90AA1HSP90AB1NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2203161-B1 QUINONE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF UNIV INDIANA RES & TECH CORP (US) 2018-05-09 EP disclosed