SCHEMBL20123554

SCHEMBL20123554

Fc1ccc2c(c1)CSc1ccccc1C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 2/20 0.43
AURKA O14965 1/20 0.38
CHEK2 O96017 1/20 0.38
CDK1 P06493 1/20 0.38
PIM1 P11309 1/20 0.38
FGFR1 P11362 1/20 0.38
CDK2 P24941 1/20 0.38
MARK3 P27448 1/20 0.38
CSNK2A1 P68400 1/20 0.38
MARK2 Q7KZI7 1/20 0.38
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
NOTUM Q6P988 1/20 0.35
NOX1 Q9Y5S8 1/20 0.34
MAPT P10636 2/20 0.34
ALDH1A1 P00352 2/20 0.33
PARP1 P09874 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20123676 0.93 HSD17B3 (0.46) HSD17B3AURKACHEK2CDK1PIM1
SCHEMBL20123579 0.88 HSD17B3 (0.47) HSD17B3AURKACHEK2CDK1PIM1
SCHEMBL20014486 0.88 HSD17B3 (0.50) HSD17B3AURKACHEK2CDK1PIM1
SCHEMBL3772410 0.81 HSD17B3 (0.43) HSD17B3NOTUMMAPTALDH1A1GAA
SCHEMBL20123505 0.80 AURKA (0.44) HSD17B3AURKACHEK2CDK1PIM1
SCHEMBL20014745 0.79 HSD17B3 (0.43) HSD17B3CA1CA2CA4CA6
SCHEMBL20014548 0.79 HPGD (0.45) HSD17B3CA1CA2CA4CA6
SCHEMBL6907006 0.79 CA1 (0.44) CA1CA2CA4CA6MAPT
SCHEMBL20014459 0.79 HSD17B3 (0.46) HSD17B3CA1CA2CA4CA6
SCHEMBL20123665 0.77 RYR2 (0.34) HSD17B3AURKACHEK2CDK1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3753936-A1 PYRIDONE DERIVATIVE, COMPOSITION THEREOF AND APPLICATION THEREOF AS ANTI-INFLUENZA DRUG Jiangxi Caishi Pharmaceutical Technology Co., Ltd. (CN) 2020-12-23 EP disclosed
EP-3428170-A1 ANTI-INFLUENZA POLYCYCLIC PYRIDONE DERIVATIVE AND PRODRUG THEREOF SHIONOGI & CO., LTD (JP) 2019-01-16 EP disclosed
EP-2620436-B1 SUBSTITUTED POLYCYCLIC CARBAMOYL PYRIDONE DERIVATIVE PRODRUG SHIONOGI & CO (JP) 2018-05-09 EP disclosed