SCHEMBL2012515

SCHEMBL2012515

CN(C(=O)c1ccc2[nH]ccc2c1)C(CCNC(=O)c1cccn1C)Cc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.65
HCRTR2 O43614 2/20 0.65
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
MAPK14 Q16539 2/20 0.39
DRD5 P21918 1/20 0.38
PADI4 Q9UM07 1/20 0.38
PADI2 Q9Y2J8 1/20 0.38
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
SLC6A3 Q01959 3/20 0.38
CTNNB1 P35222 1/20 0.37
WNT3A P56704 1/20 0.37
HDAC1 Q13547 3/20 0.37
HDAC2 Q92769 3/20 0.37
HDAC3 O15379 2/20 0.37
HDAC4 P56524 2/20 0.37
HDAC7 Q8WUI4 2/20 0.37
HDAC10 Q969S8 2/20 0.37
HDAC8 Q9BY41 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012583 0.87 HCRTR1 (0.64) HCRTR1HCRTR2NPC1RAB9ACTNNB1
SCHEMBL2014120 0.85 HCRTR1 (0.68) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2017845 0.85 HCRTR1 (0.68) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2010943 0.85 HCRTR1 (0.66) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL13139060 0.85 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2010961 0.84 HCRTR1 (0.64) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2015169 0.83 HCRTR1 (0.65) HCRTR1HCRTR2NPC1RAB9AMAPK14
SCHEMBL2011913 0.83 HCRTR1 (0.45) HCRTR1HCRTR2NPC1RAB9AMAPK14
SCHEMBL2011909 0.83 HCRTR1 (0.45) HCRTR1HCRTR2NPC1RAB9AMAPK14
SCHEMBL2013785 0.83 HCRTR1 (0.67) HCRTR1HCRTR2NPC1RAB9APADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed