SCHEMBL20125424

SCHEMBL20125424

C=C(/C=C\C)N1CCCC(NC)C1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 6/20 0.35
JAK1 P23458 1/20 0.35
CA1 P00915 4/20 0.34
CA2 P00918 4/20 0.34
CA12 O43570 2/20 0.34
CA9 Q16790 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14457193 0.78 CA1 (0.38) CA1CA2CA12CA9
SCHEMBL13328191 0.73 CA1 (0.36) CA1CA2CA12CA9
SCHEMBL17378886 0.72
SCHEMBL19909890 0.72 KDM4E (0.31)
SCHEMBL19240692 0.72 JAK3 (0.49) JAK3JAK1
SCHEMBL19240687 0.72 JAK3 (0.49) JAK3JAK1
SCHEMBL19240693 0.72 JAK3 (0.49) JAK3JAK1
SCHEMBL28206408 0.72 CA1 (0.46) CA1CA2CA12CA9
SCHEMBL24244429 0.71 JAK3 (0.48) JAK3CA1CA2CA12CA9
SCHEMBL20962117 0.70 ALDH1A1 (0.33) CA1CA2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3318565-A1 PYRROLO[2,3-D]PYRIMIDINYL, PYRROLO[2,3-B]PYRAZINYL AND PYRROLO[2,3-D]PYRIDINYL ACRYLAMIDES Pfizer Inc (US) 2018-05-09 EP disclosed