SCHEMBL2013118

SCHEMBL2013118

CCCC(C)(C)c1cc(Nc2ccccc2)ccc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 11/20 0.41
GAA P10253 6/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
TDP1 Q9NUW8 3/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 2/20 0.41
GFER P55789 1/20 0.41
ALDH1A1 P00352 9/20 0.41
ALOX12 P18054 4/20 0.41
CYP3A4 P08684 4/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2C19 P33261 3/20 0.41
HTT P42858 1/20 0.41
AR P10275 1/20 0.39
HSD17B10 Q99714 3/20 0.38
ALOX15 P16050 2/20 0.38
MAPK1 P28482 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21634341 0.92 MAPT (0.39) MAPTGAAMEN1KMT2ATDP1
SCHEMBL26114037 0.81 MAPT (0.48) MAPTGAAMEN1KMT2ATDP1
SCHEMBL28021914 0.77 MAPT (0.39) MAPTGAAMEN1KMT2ATDP1
SCHEMBL886922 0.75 GAA (0.50) MAPTGAAMEN1KMT2ATDP1
SCHEMBL8160618 0.74 GAA (0.37) MAPTGAAMEN1KMT2AKDM4E
SCHEMBL27518609 0.73 MAPT (0.42) MAPTGAAMEN1KMT2ATDP1
SCHEMBL6470377 0.73 CNR1 (0.38) MAPTGAAMEN1KMT2ATDP1
SCHEMBL536379 0.72 MAPT (0.46) MAPTGAAMEN1KMT2ATDP1
SCHEMBL5613090 0.72 MAPT (0.49) MAPTGAAMEN1KMT2ATDP1
SCHEMBL3796679 0.71 MAPT (0.48) MAPTGAAMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 168 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101641402-A Tire rubber composition containing a novel antioxidant system MICHELIN SOC TECH FR 2010-02-03 CN claimed
EP-1027327-A4 FORMATION OF QUINONEDIIMINES FROM PHENYLENEDIAMINES BY CATALYTIC OXIDATION FLEXSYS AMERICA LP (US) 2000-11-29 EP claimed
EP-1027327-A1 FORMATION OF QUINONEDIIMINES FROM PHENYLENEDIAMINES BY CATALYTIC OXIDATION FLEXSYS AMERICA L.P. (US) 2000-08-16 EP claimed
WO-1999021827-A1 FORMATION OF QUINONEDIIMINES FROM PHENYLENEDIAMINES BY CATALYTIC OXIDATION FLEXSYS AMERICA L.P. (US) 1999-05-06 WO claimed
WO-2024145438-A1 CURED EPOXY RESIN AND METHOD OF CURING AN EPOXY RESIN USING AN AMINE COMPOUND SI GROUP, INC. (US) 2024-07-04 WO disclosed
CN-118032800-A Terahertz Characterization of Multi-Layer Tire Tread 固特异轮胎和橡胶公司 2024-05-14 CN disclosed
CN-114829478-B Elastomer composition reinforced by ground biochar 米其林集团总公司 2024-04-16 CN disclosed
US-20240102926-A1 TERAHERTZ CHARACTERIZATION OF A MULTI-LAYERED TIRE TREAD THE GOODYEAR TIRE & RUBBER COMPANY 2024-03-28 US disclosed
EP-4331821-A1 METHOD AND APPARATUS FOR TERAHERTZ CHARACTERIZATION OF A MULTI-LAYERED TIRE TREAD The Goodyear Tire & Rubber Company (US) 2024-03-06 EP disclosed
US-11874223-B1 Terahertz characterization of a multi-layered tire tread THE GOODYEAR TIRE & RUBBER COMPANY (US) 2024-01-16 US disclosed
EP-4061645-A1 RUBBER COMPOSITION INCLUDING A FUNCTIONALISED POLYBUTADIENE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2022-09-28 EP disclosed
CN-114829478-A Elastomer composition reinforced by ground biochar 米其林集团总公司 2022-07-29 CN disclosed
US-6182728-B1 Pneumatic run flat tire HANKOOK TIRE 2001-02-06 US disclosed
EP-0649446-B1 METHOD AND COMPOSITION FOR USING SUBSTITUTED MELAMINES AS NOVOLAK RESIN CURING AGENTS MICHELIN & CIE (FR) 1999-12-15 EP disclosed
WO-1999062868-A1 PREPARATION OF QUINONEDIIMINES FROM PHENYLENEDIAMINES USING OXYGEN AND A METAL OR METAL SALT CATALYST FLEXSYS AMERICA L.P. (US) 1999-12-09 WO disclosed
EP-0649446-A1 METHOD AND COMPOSITION FOR USING SUBSTITUTED MELAMINES AS NOVOLAK RESIN CURING AGENTS COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN-MICHELIN & CIE (FR) 1995-04-26 EP disclosed
WO-1994001493-A1 METHOD AND COMPOSITION FOR USING SUBSTITUTED MELAMINES AS NOVOLAK RESIN CURING AGENTS COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN - MICHELIN & CIE (FR) 1994-01-20 WO disclosed
US-4396052-A SANDWICH LAYER OF VULCANIZED BLENDS OF 1,3-BUTADIENE-METHYLALLENE POLYMER AND NATURAL RUBBER OR POLYISOPRENE THE YOKOHAMA RUBBER CO., LTD. (JP) 1983-08-02 US disclosed
US-4347290-A HAVING AN ADHESIVE COATING OF A BRASS ALLOY CONTAINING COBALT N.V. BEKAERT S.A. (BE) 1982-08-31 US disclosed
US-4255496-A Steel wire reinforcing elements with a brass-cobalt alloy adhesive coating N. V. BEKAERT S.A. (BE) 1981-03-10 US disclosed