SCHEMBL2013232

SCHEMBL2013232

Cc1nc2ccc(C(=O)N(C)C(CCNC(=O)c3cccn3C)Cc3ccccc3)cc2o1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.63
HCRTR2 O43614 2/20 0.63
TP53 P04637 6/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
LMNA P02545 2/20 0.43
MME P08473 1/20 0.43
TAS1R3 Q7RTX0 3/20 0.41
TAS1R1 Q7RTX1 3/20 0.41
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2010621 0.94 HCRTR1 (0.63) HCRTR1HCRTR2TP53NPC1RAB9A
SCHEMBL2014534 0.86 HCRTR1 (0.66) HCRTR1HCRTR2TP53NPC1RAB9A
SCHEMBL2013109 0.85 HCRTR1 (0.64) HCRTR1HCRTR2TP53NPC1RAB9A
SCHEMBL2015002 0.85 HCRTR1 (0.69) HCRTR1HCRTR2TP53NPC1RAB9A
SCHEMBL2010631 0.85 HCRTR1 (0.65) HCRTR1HCRTR2TP53NPC1RAB9A
SCHEMBL2013242 0.84 HCRTR1 (0.70) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL2015950 0.84 HCRTR1 (0.70) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL2012339 0.84 HCRTR1 (0.63) HCRTR1HCRTR2TP53NPC1RAB9A
SCHEMBL2011910 0.84 HCRTR1 (0.69) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL2013785 0.84 HCRTR1 (0.67) HCRTR1HCRTR2NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed