SCHEMBL20132369

SCHEMBL20132369

C[C@H](Nc1ccc(C(=O)NO)nc1)c1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 16/20 0.65
HDAC1 Q13547 16/20 0.65
HDAC6 Q9UBN7 11/20 0.65
HDAC8 Q9BY41 8/20 0.65
HDAC4 P56524 7/20 0.65
HDAC2 Q92769 7/20 0.59
KDM4E B2RXH2 1/20 0.50
ASPH Q12797 1/20 0.50
RIOX2 Q8IUF8 1/20 0.50
KDM8 Q8N371 1/20 0.50
NCOR2 Q9Y618 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26697537 1.00 HDAC3 (0.65) HDAC3HDAC1HDAC6HDAC8HDAC4
SCHEMBL20132370 1.00 HDAC3 (0.65) HDAC3HDAC1HDAC6HDAC8HDAC4
SCHEMBL20132421 0.86 HDAC1 (0.61) HDAC3HDAC1HDAC6HDAC8HDAC4
SCHEMBL20142362 0.83 KDM4E (0.50) HDAC3HDAC1HDAC6HDAC8HDAC4
SCHEMBL21226799 0.83 KDM4E (0.50) HDAC3HDAC1HDAC6HDAC8HDAC4
SCHEMBL20132427 0.83 KDM4E (0.50) HDAC3HDAC1HDAC6HDAC8HDAC4
SCHEMBL11399034 0.76 P4HTM (0.56) KDM4EASPHRIOX2KDM8
SCHEMBL20161299 0.75 HDAC3 (0.49) HDAC3HDAC1HDAC6HDAC8HDAC4
SCHEMBL8738685 0.74 HDAC6 (1.00) HDAC3HDAC1HDAC6HDAC2
SCHEMBL4730094 0.74 HDAC6 (1.00) HDAC3HDAC1HDAC6HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538084-B1 PHENYL AND PYRIDINYL HYDROXAMIC ACIDS ACETYLON PHARMACEUTICALS INC (US) 2023-11-01 EP disclosed
US-10927072-B2 Phenyl and pyridinyl hydroxamic acids ACETYLON PHARMACEUTICALS, INC. (US) 2021-02-23 US disclosed
US-10370324-B2 Phenyl and pyridinyl hydroxamic acids ACETYLON PHARMACEUTICALS, INC. (US) 2019-08-06 US disclosed
US-20180127356-A1 PHENYL AND PYRIDINYL HYDROXAMIC ACIDS ACETYLON PHARMACEUTICALS, INC. 2018-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10370324-B2 Phenyl and pyridinyl hydroxamic acids HDAC6, HDAC1, HDAC5 HDAC3 4/4885HDAC1 2/4885HDAC6 1/4885
US-10927072-B2 Phenyl and pyridinyl hydroxamic acids HDAC6, HDAC1, HDAC5 HDAC3 4/4885HDAC1 2/4885HDAC6 1/4885
US-20180127356-A1 PHENYL AND PYRIDINYL HYDROXAMIC ACIDS HDAC6, HDAC1, HDAC5 HDAC3 4/4885HDAC1 2/4885HDAC6 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.