SCHEMBL20135491

SCHEMBL20135491

C[Si](C)(C)CCOCn1nc(C2CCN(C(=O)O)CC2)c2c(Br)cc(Br)cc21

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 2/20 0.33
EPHX2 P34913 1/20 0.31
P2RX7 Q99572 1/20 0.30
NPC1 O15118 1/20 0.30
DGAT1 O75907 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29688849 0.88 CNR1 (0.41)
SCHEMBL20134963 0.88 CNR1 (0.41)
SCHEMBL20135277 0.80 CNR1 (0.40) DGAT1
SCHEMBL17844426 0.76 KLKB1 (0.34) KLKB1P2RX7NPC1DGAT1
SCHEMBL17844574 0.74 CHRM4 (0.35) KLKB1DGAT1
SCHEMBL20135368 0.73 CNR1 (0.41) EPHX2
SCHEMBL17844648 0.72 NPC1 (0.36) KLKB1P2RX7NPC1DGAT1
SCHEMBL20135506 0.71 CNR1 (0.41)
SCHEMBL28672490 0.70 PIM1 (0.30)
SCHEMBL492579 0.70 F2RL1 (0.34) KLKB1NPC1DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3321256-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE Mitsubishi Tanabe Pharma Corporation (JP) 2018-05-16 EP disclosed