SCHEMBL17844648

SCHEMBL17844648

C[Si](C)(C)CCOCn1nc(C2CCN(C(=O)O)CC2)c2cccnc21

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
CFD P00746 2/20 0.35
CHRM4 P08173 2/20 0.35
CHRM2 P08172 1/20 0.34
CHRNA7 P36544 1/20 0.34
P2RX7 Q99572 1/20 0.34
KLKB1 P03952 1/20 0.33
HTR3A P46098 2/20 0.33
HSD11B1 P28845 2/20 0.33
CNR1 P21554 2/20 0.33
CNR2 P34972 2/20 0.33
DGAT1 O75907 1/20 0.33
ELANE P08246 1/20 0.32
REN P00797 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17838312 0.88 CNR1 (0.43) CNR1
SCHEMBL17844426 0.84 KLKB1 (0.34) NPC1CHRM4CHRM2CHRNA7P2RX7
SCHEMBL17844574 0.82 CHRM4 (0.35) CHRM4CHRM2KLKB1DGAT1
SCHEMBL16516469 0.77 CFD (0.40) NPC1CFDHTR3ACNR1CNR2
SCHEMBL23163208 0.75 CFD (0.43) NPC1CFD
SCHEMBL30092705 0.74 CFD (0.50) NPC1CFDHTR3ACNR1CNR2
SCHEMBL16532464 0.73 CFD (0.41) NPC1CFDHTR3ACNR1CNR2
SCHEMBL17837846 0.73 HPGD (0.40) CNR1
SCHEMBL29900927 0.73 CNR1 (0.43) KLKB1CNR1
SCHEMBL20135491 0.72 KLKB1 (0.33) NPC1P2RX7KLKB1DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233829-A1 PYRIMIDINE AND TRIAZINE DERIVATIVES AND THEIR USE AS AXL INHIBITORS Pfizer Inc (US) 2017-10-25 EP disclosed
WO-2016097918-A1 PYRIMIDINE AND TRIAZINE DERIVATIVES AND THEIR USE AS AXL INHIBITORS PFIZER INC. (US) 2016-06-23 WO disclosed