SCHEMBL20135909

SCHEMBL20135909

Cc1c[c]c(-c2ncccn2)nc1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28362084 0.80
SCHEMBL28361818 0.77 KDM4E (0.45) CCR1CCR5CCR8
SCHEMBL28361794 0.76 CYP2A6 (0.46) CCR1CCR5CCR8
SCHEMBL28051848 0.69 PDPK1 (0.36)
SCHEMBL193940 0.67
SCHEMBL1672214 0.67 ALDH1A1 (0.34)
SCHEMBL1671362 0.66 CYP2A6 (0.30)
SCHEMBL28358273 0.65 CCR1 (0.38) CCR1CCR5CCR8
SCHEMBL790783 0.64
SCHEMBL9098711 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP claimed
CN-110669052-B Substituted 2-azabicyclic compounds and their use as orexin receptor modulators 詹森药业有限公司 2022-10-11 CN disclosed
CN-110669052-A Substituted 2-azabicyclic compounds and their use as orexin receptor modulators 詹森药业有限公司 2020-01-10 CN disclosed