SCHEMBL2013816

SCHEMBL2013816

CN(C(=O)c1ccc2[nH]ccc2c1)C(CCNC(=O)c1nc2ccccc2n1C)Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.45
HCRTR2 O43614 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
MAPK14 Q16539 2/20 0.37
DRD5 P21918 1/20 0.36
KLK5 Q9Y337 1/20 0.36
PADI4 Q9UM07 1/20 0.36
PADI2 Q9Y2J8 1/20 0.36
GAA P10253 1/20 0.36
NAMPT P43490 2/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
RECQL P46063 1/20 0.35
NFATC1 O95644 1/20 0.35
CTNNB1 P35222 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13139041 1.00 HCRTR1 (0.45) HCRTR1HCRTR2SMN1; SMN2NPC1TP53
SCHEMBL13138975 0.89 HCRTR1 (0.50) HCRTR1HCRTR2SMN1; SMN2NPC1TP53
SCHEMBL13138972 0.87 HCRTR1 (0.50) HCRTR1HCRTR2SMN1; SMN2NPC1TP53
SCHEMBL2015176 0.84 HCRTR1 (0.40) HCRTR1HCRTR2SMN1; SMN2NPC1TP53
SCHEMBL13138938 0.84 HCRTR1 (0.40) HCRTR1HCRTR2SMN1; SMN2NPC1TP53
SCHEMBL13139038 0.84 HCRTR1 (0.48) HCRTR1HCRTR2SMN1; SMN2NPC1TP53
SCHEMBL13139073 0.84 HCRTR1 (0.53) HCRTR1HCRTR2SMN1; SMN2NPC1TP53
SCHEMBL13139051 0.83 HCRTR1 (0.47) HCRTR1HCRTR2SMN1; SMN2NPC1TP53
SCHEMBL13138966 0.83 HCRTR1 (0.45) HCRTR1HCRTR2SMN1; SMN2NPC1TP53
SCHEMBL13138988 0.83 GAA (0.47) HCRTR1HCRTR2SMN1; SMN2NPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed