SCHEMBL2015176

SCHEMBL2015176

CN(C(=O)c1cccc2[nH]ccc12)C(CCNC(=O)c1nc2ccccc2n1C)Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.40
HCRTR2 O43614 2/20 0.40
HPGDS O60760 1/20 0.35
PDE10A Q9Y233 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC2 Q92769 2/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK14 Q16539 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
TSHR P16473 1/20 0.35
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13138938 1.00 HCRTR1 (0.40) HCRTR1HCRTR2HPGDSPDE10ASMN1; SMN2
SCHEMBL13138950 0.89 HCRTR1 (0.43) HCRTR1HCRTR2PDE10ASMN1; SMN2ALDH1A1
SCHEMBL6919279 0.86 HCRTR1 (0.45) HCRTR1HCRTR2PDE10ASMN1; SMN2HDAC1
SCHEMBL13139041 0.84 HCRTR1 (0.45) HCRTR1HCRTR2SMN1; SMN2MAPK14NPC1
SCHEMBL2013191 0.84 HCRTR1 (0.40) HCRTR1HCRTR2PDE10ASMN1; SMN2ALDH1A1
SCHEMBL2013816 0.84 HCRTR1 (0.45) HCRTR1HCRTR2SMN1; SMN2MAPK14NPC1
SCHEMBL6917383 0.84 HCRTR1 (0.40) HCRTR1HCRTR2PDE10ASMN1; SMN2ALDH1A1
SCHEMBL13138972 0.83 HCRTR1 (0.50) HCRTR1HCRTR2PDE10ASMN1; SMN2ALDH1A1
SCHEMBL13138955 0.83 GAA (0.42) HCRTR1HCRTR2PDE10ASMN1; SMN2TSHR
SCHEMBL13138957 0.83 C5AR1 (0.41) HCRTR1HCRTR2PDE10ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed