SCHEMBL20138480

SCHEMBL20138480

c1ccc(CCc2ncc3ccsc3n2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.44
PIN1 Q13526 1/20 0.43
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4C Q08493 2/20 0.42
PDE4D Q08499 2/20 0.42
PLA2G4A P47712 1/20 0.38
NOS1 P29475 1/20 0.38
KCNH2 Q12809 1/20 0.38
CES1 P23141 1/20 0.38
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
PKM P14618 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20631751 0.78 HRH1 (0.30)
SCHEMBL28654885 0.76 PDE4A (0.50) HTR2CPIN1PDE4APDE4BPDE4C
SCHEMBL12343963 0.74 ADORA2A (0.37) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL5439409 0.74 CYP2A6 (0.35)
SCHEMBL27374635 0.73 HTR2C (0.49) HTR2CPIN1PDE4APDE4BPDE4C
SCHEMBL30918003 0.73 HTR2C (0.49) HTR2CPIN1PDE4APDE4BPDE4C
SCHEMBL14964889 0.71 HRH3 (0.39) TDP1L3MBTL1
SCHEMBL19838265 0.70
SCHEMBL14965474 0.69 ADORA2A (0.51) MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL19714623 0.68 HTR2C (0.48) HTR2CPIN1NOS1KCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180132516-A1 POSITIVE ALLOSTERIC MODULATORS OF SWEET TASTE SENSORYGEN INC (US) 2018-05-17 US disclosed