SCHEMBL20139031

SCHEMBL20139031

C=CC(=O)Nc1cccc(Nc2ncnc3[nH]c(-c4cnn(C)c4)cc23)c1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.57
JAK3 P52333 2/20 0.57
JAK1 P23458 1/20 0.55
RET P07949 2/20 0.54
SRC P12931 1/20 0.52
AURKB Q96GD4 10/20 0.51
AURKA O14965 1/20 0.51
KIT P10721 1/20 0.51
FLT3 P36888 1/20 0.51
BTK Q06187 2/20 0.51
EGFR P00533 3/20 0.50
PIK3CD O00329 1/20 0.50
ERBB2 P04626 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20150470 0.85 EGFR (0.57) JAK2JAK3BTKEGFRERBB2
SCHEMBL20139048 0.85 SRC (0.59) JAK3JAK1SRCBTKEGFR
SCHEMBL20143667 0.84 PIK3CD (0.56) JAK3SRCBTKEGFRPIK3CD
SCHEMBL21484334 0.83 ERBB2 (0.62) JAK2JAK3SRCEGFRERBB2
SCHEMBL20138979 0.83 BTK (0.54) JAK3SRCKITBTKEGFR
SCHEMBL20139785 0.81 SRC (0.58) SRCBTKEGFRPIK3CDERBB2
SCHEMBL20139002 0.80 PIK3CD (0.55) JAK3SRCBTKEGFRPIK3CD
SCHEMBL20150708 0.80 PIK3CD (0.54) JAK3SRCBTKEGFRPIK3CD
SCHEMBL29538618 0.80 JAK1 (0.59) JAK2JAK3JAK1BTKEGFR
SCHEMBL20139429 0.80 JAK1 (0.59) JAK2JAK3JAK1BTKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018088780-A1 NOVEL PYRROLOPYRIMIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2018-05-17 WO disclosed