SCHEMBL20139625

SCHEMBL20139625

C[C@@]1(c2ccc(F)cc2)CNC[C@@H]1c1cc(F)c(-c2ccccc2)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.48
NR1I2 O75469 1/20 0.48
DRD1 P21728 2/20 0.39
NPY5R Q15761 1/20 0.34
CHRNA1 P02708 2/20 0.33
CHRNG P07510 2/20 0.33
CHRNB1 P11230 2/20 0.33
CHRNB2 P17787 2/20 0.33
SLC6A2 P23975 2/20 0.33
CHRNB4 P30926 2/20 0.33
CHRNA3 P32297 2/20 0.33
CHRNA4 P43681 2/20 0.33
CHRND Q07001 2/20 0.33
SLC6A3 Q01959 1/20 0.33
KDM1A O60341 1/20 0.32
RCOR1 Q9UKL0 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139590 1.00 RORC (0.48) RORCNR1I2DRD1NPY5RCHRNA1
SCHEMBL20139610 0.86 RORC (0.57) RORCNR1I2DRD1NPY5RCHRNA1
SCHEMBL20139691 0.86 RORC (0.57) RORCNR1I2DRD1NPY5RCHRNA1
SCHEMBL20149299 0.84 RORC (0.51) RORCNR1I2DRD1CHRNA1CHRNG
SCHEMBL20139577 0.84 RORC (0.51) RORCNR1I2DRD1CHRNA1CHRNG
SCHEMBL20139575 0.84 RORC (0.51) RORCNR1I2DRD1CHRNA1CHRNG
Trifluoroacetic Acid SCHEMBL20139646 0.78 RORC (0.52) RORCNR1I2SLC6A2SLC6A3
Trifluoroacetic Acid SCHEMBL20139647 0.78 RORC (0.52) RORCNR1I2SLC6A2SLC6A3
SCHEMBL23713083 0.77 RORC (0.46) RORCNR1I2DRD1
SCHEMBL20139645 0.72 RORC (0.55) RORCNR1I2SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538522-A1 ROR GAMMA MODULATORS Bristol-Myers Squibb Company (US) 2019-09-18 EP disclosed
WO-2018089406-A1 ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed