SCHEMBL20139802

SCHEMBL20139802

Cc1ccc2c(C#N)nn(Cc3cccc(F)c3F)c2n1.N#Cc1nn(Cc2ccccc2F)c2nccnc12

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 18/20 0.44
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16370341 0.88 PDE5A (0.52) PDE5ATDP1L3MBTL1ADORA2AADORA1
SCHEMBL20140367 0.86 TDP1 (0.45) PDE5ATDP1L3MBTL1ADORA2AADORA1
SCHEMBL21775364 0.83 ALDH1A1 (0.41) PDE5AADORA2AADORA1
SCHEMBL2881224 0.78 PDE5A (0.42) PDE5AL3MBTL1
SCHEMBL15111735 0.76 PDE5A (0.55) PDE5AADORA2AADORA1
SCHEMBL16370487 0.76 PDE5A (0.53) PDE5AADORA2AADORA1
SCHEMBL174888 0.76 PDE5A (0.48) PDE5A
SCHEMBL30745084 0.76 PDE5A (0.48) PDE5A
SCHEMBL14746447 0.74 PDE5A (0.54) PDE5ATDP1L3MBTL1ADORA2AADORA1
SCHEMBL14746488 0.74 PDE5A (0.52) PDE5ATDP1L3MBTL1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538520-A2 SGC STIMULATORS Cyclerion Therapeutics, Inc. (US) 2019-09-18 EP disclosed
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed