SCHEMBL20140062

SCHEMBL20140062

COc1ccc([C@H](CC(=O)O)N2C[C@](C)(CCCCC(C)=O)C2=O)cn1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 14/20 0.46
ITGB3 P05106 13/20 0.46
ITGB1 P05556 3/20 0.43
ITGB6 P18564 3/20 0.43
ITGA2B P08514 3/20 0.43
ITGA5 P08648 2/20 0.43
ITGB8 P26012 2/20 0.43
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
HSD11B1 P28845 1/20 0.34
ITGA4 P13612 1/20 0.34
FFAR1 O14842 1/20 0.34
ITGB5 P18084 1/20 0.34
P2RX3 P56373 1/20 0.33
P2RX2 Q9UBL9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21314474 1.00 ITGAV (0.46) ITGAVITGB3ITGB1ITGB6ITGA2B
SCHEMBL21314477 1.00 ITGAV (0.46) ITGAVITGB3ITGB1ITGB6ITGA2B
SCHEMBL28744049 0.89 ITGB3 (0.37) ITGAVITGB3ITGB1ITGB6ITGA2B
SCHEMBL30487525 0.89 ITGB3 (0.37) ITGAVITGB3ITGB1ITGB6ITGA2B
SCHEMBL20158223 0.89 ITGB3 (0.37) ITGAVITGB3ITGB1ITGB6ITGA2B
SCHEMBL21314435 0.87 ITGAV (0.43) ITGAVITGB3ITGB1ITGB6ITGA2B
SCHEMBL21314434 0.87 ITGAV (0.43) ITGAVITGB3ITGB1ITGB6ITGA2B
SCHEMBL20140498 0.87 ITGAV (0.43) ITGAVITGB3ITGB1ITGB6ITGA2B
SCHEMBL20140602 0.87 ITGAV (0.43) ITGAVITGB3ITGB1ITGB6ITGA2B
SCHEMBL20141198 0.84 ITGAV (0.48) ITGAVITGB3ITGB1ITGB6ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538526-A1 CYCLOBUTANE- AND AZETIDINE-CONTAINING MONO AND SPIROCYCLIC COMPOUNDS AS ALPHA V INTEGRIN INHIBITORS Bristol-Myers Squibb Company (US) 2019-09-18 EP disclosed
WO-2018089355-A1 CYCLOBUTANE- AND AZETIDINE-CONTAINING MONO AND SPIROCYCLIC COMPOUNDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed