SCHEMBL20140217

SCHEMBL20140217

COc1ccc(C(CC(=O)O)c2nc(CCCc3ccc4cccnc4n3)co2)cc1F

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.41
ITGAV P06756 2/20 0.41
ITGA2B P08514 1/20 0.41
ITGB6 P18564 1/20 0.41
CTSA P10619 11/20 0.39
SUCNR1 Q9BXA5 7/20 0.38
BDKRB1 P46663 1/20 0.38
OXGR1 Q96P68 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142767 0.92 ITGB3 (0.40) ITGB3ITGAVITGA2BITGB6SUCNR1
SCHEMBL29797239 0.92 ITGB3 (0.40) ITGB3ITGAVITGA2BITGB6SUCNR1
SCHEMBL20141912 0.80 CTSA (0.38) ITGB3ITGAVITGA2BITGB6CTSA
SCHEMBL21294620 0.80 CTSA (0.38) ITGB3ITGAVITGA2BITGB6CTSA
SCHEMBL20140302 0.79 ITGB3 (0.38) ITGB3ITGAVITGA2BITGB6SUCNR1
SCHEMBL20140538 0.79 ITGAV (0.65) ITGB3ITGAVITGA2BITGB6
SCHEMBL20139938 0.79 ITGAV (0.65) ITGB3ITGAVITGA2BITGB6
SCHEMBL20139714 0.79 ITGAV (0.65) ITGB3ITGAVITGA2BITGB6
SCHEMBL21311604 0.79 SUCNR1 (0.38) ITGB3ITGAVITGA2BITGB6CTSA
SCHEMBL20139608 0.78 ITGB3 (0.40) ITGB3ITGAVITGA2BITGB6CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538525-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS Bristol-Myers Squibb Company (US) 2019-09-18 EP disclosed
WO-2018089353-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed