SCHEMBL20140559

SCHEMBL20140559

Cc1ccccc1N1CCN(Cc2cc(C(=O)N3CCN(c4ccccc4)CC3)n(C)c2)CC1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.52
RPTOR Q8N122 2/20 0.52
MLST8 Q9BVC4 2/20 0.52
HRH3 Q9Y5N1 2/20 0.51
ATM Q13315 1/20 0.50
HTR7 P34969 2/20 0.48
DRD2 P14416 1/20 0.48
HTR2A P28223 1/20 0.48
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TSHR P16473 1/20 0.46
MYC P01106 1/20 0.45
AR P10275 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158933 0.90 HRH3 (0.47) MTORRPTORMLST8HRH3ATM
SCHEMBL20159024 0.90 MTOR (0.64) MTORRPTORMLST8HRH3HTR7
SCHEMBL20159166 0.89 POLB (0.55) MTORRPTORMLST8HRH3HTR7
SCHEMBL20159007 0.89 POLB (0.55) MTORRPTORMLST8HRH3HTR7
SCHEMBL20159123 0.87 MTOR (0.69) MTORRPTORMLST8HRH3HTR7
SCHEMBL20158948 0.86 MTOR (0.49) MTORRPTORMLST8HRH3HTR7
SCHEMBL20159115 0.82 MTOR (0.55) MTORRPTORMLST8HRH3HTR7
SCHEMBL20159302 0.80 TP53 (0.53) DRD2HTR2AMEN1KMT2AALDH1A1
SCHEMBL20159079 0.80 MTOR (0.52) MTORRPTORMLST8HRH3HTR7
SCHEMBL20159286 0.79 MTOR (0.51) MTORRPTORMLST8HRH3HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed