SCHEMBL20140701

SCHEMBL20140701

C[C@H]1CN(c2cc(F)c(C#N)cc2F)CCN1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
LMNA P02545 1/20 0.39
CHRM2 P08172 1/20 0.39
HTR2C P28335 1/20 0.38
USP28 Q96RU2 2/20 0.36
USP25 Q9UHP3 1/20 0.36
TRPV4 Q9HBA0 1/20 0.36
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
MAPT P10636 1/20 0.34
AKR1B1 P15121 1/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
AXL P30530 1/20 0.33
FLT3 P36888 1/20 0.33
TYRO3 Q06418 1/20 0.33
MERTK Q12866 1/20 0.33
PMP22 Q01453 1/20 0.33
ALK Q9UM73 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20141175 0.90 ALDH1A1 (0.45) ALDH1A1LMNAHTR2CUSP28USP25
SCHEMBL12182701 0.81 ALDH1A1 (0.44) ALDH1A1LMNACHRM2HTR2CALK
SCHEMBL12182668 0.81 ALDH1A1 (0.44) ALDH1A1LMNACHRM2HTR2CALK
Hydrochloric Acid SCHEMBL29767487 0.80 ALDH1A1 (0.46) ALDH1A1LMNACHRM2HTR2CALK
Hydrochloric Acid SCHEMBL28829934 0.80 ALDH1A1 (0.46) ALDH1A1LMNACHRM2HTR2CALK
Hydrochloric Acid SCHEMBL28829935 0.80 ALDH1A1 (0.46) ALDH1A1LMNACHRM2HTR2CALK
SCHEMBL20159179 0.80 ALDH1A1 (0.43) ALDH1A1LMNAHTR2CKCNH2HRH3
SCHEMBL18825914 0.80 KHK (0.46) ALDH1A1CHRM2KCNH2MAPTBCL2A1
SCHEMBL8295259 0.79 ALDH1A1 (0.75) ALDH1A1LMNAUSP28USP25TRPV4
SCHEMBL30073656 0.79 ALDH1A1 (0.75) ALDH1A1LMNAUSP28USP25TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed