SCHEMBL20140792

SCHEMBL20140792

CN(C)C(=O)c1ccc(C(CC(=O)O)c2nc(CCCCC3CCc4cccnc4N3)cs2)cc1F

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 16/20 0.36
ITGB3 P05106 15/20 0.36
ITGB6 P18564 10/20 0.36
ITGA2B P08514 7/20 0.36
ITGB5 P18084 4/20 0.33
CTSA P10619 1/20 0.32
ITGB8 P26012 3/20 0.31
NQO1 P15559 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
IDH1 O75874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140148 0.85 ITGB3 (0.47) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL20141460 0.80 ITGAV (0.57) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL20153423 0.80 ITGAV (0.57) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL29797098 0.80 ITGAV (0.57) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL29797207 0.80 ITGAV (0.57) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL20140790 0.80 ITGAV (0.57) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL21294589 0.79 ITGB3 (0.47) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL21294608 0.79 ITGB3 (0.47) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL21294590 0.79 ITGB3 (0.47) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL20139506 0.79 ITGB3 (0.47) ITGAVITGB3ITGB6ITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538525-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS Bristol-Myers Squibb Company (US) 2019-09-18 EP claimed
WO-2018089353-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO claimed