SCHEMBL20141855

SCHEMBL20141855

O=C(O)C[C@H](NC(=O)CC1CN(CCCc2ccc3c(n2)NCCC3)C1)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 20/20 0.73
ITGAV P06756 20/20 0.73
ITGB5 P18084 16/20 0.73
ITGB6 P18564 16/20 0.73
ITGB8 P26012 16/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20141300 0.88 ITGAV (0.68) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20141298 0.88 ITGAV (0.68) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20157744 0.85 ITGAV (0.69) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL27132661 0.84 ITGAV (0.66) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL29162823 0.84 ITGAV (0.66) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL27003189 0.84 ITGAV (0.66) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20141596 0.84 ITGAV (0.68) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20141599 0.84 ITGAV (0.68) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL21317464 0.83 ITGAV (0.66) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20142624 0.83 ITGB3 (0.66) ITGB3ITGAVITGB5ITGB6ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538526-A1 CYCLOBUTANE- AND AZETIDINE-CONTAINING MONO AND SPIROCYCLIC COMPOUNDS AS ALPHA V INTEGRIN INHIBITORS Bristol-Myers Squibb Company (US) 2019-09-18 EP claimed
WO-2018089355-A1 CYCLOBUTANE- AND AZETIDINE-CONTAINING MONO AND SPIROCYCLIC COMPOUNDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO claimed