SCHEMBL20142712

SCHEMBL20142712

N#Cc1cccc(N2CCCCC2)c1N

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
KDM4E B2RXH2 2/20 0.50
KEAP1 Q14145 1/20 0.50
AR P10275 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
MAPT P10636 2/20 0.45
POLB P06746 1/20 0.45
HRH3 Q9Y5N1 1/20 0.44
HTT P42858 1/20 0.42
LMNA P02545 1/20 0.42
MMP1 P03956 1/20 0.42
ROCK2 O75116 2/20 0.41
ROCK1 Q13464 2/20 0.41
CDC42BPA Q5VT25 2/20 0.41
CDC42BPB Q9Y5S2 2/20 0.41
MAPK1 P28482 1/20 0.41
CSF1R P07333 1/20 0.40
NPC1 O15118 1/20 0.40
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31388194 0.83 AR (0.62) ALDH1A1KDM4EKEAP1ARL3MBTL1
SCHEMBL7524105 0.83 AR (0.62) ALDH1A1KDM4EKEAP1ARL3MBTL1
SCHEMBL7528396 0.83 AR (0.62) ALDH1A1KDM4EKEAP1ARL3MBTL1
SCHEMBL1660394 0.83 AR (0.62) ALDH1A1KDM4EKEAP1ARL3MBTL1
SCHEMBL1871089 0.82 ALDH1A1 (0.67) ALDH1A1KDM4EKEAP1ARL3MBTL1
SCHEMBL573134 0.82 ALDH1A1 (0.67) ALDH1A1KDM4EKEAP1ARL3MBTL1
SCHEMBL829177 0.81 AR (0.65) ALDH1A1KDM4EKEAP1ARL3MBTL1
SCHEMBL1878340 0.80 ALDH1A1 (0.69) ALDH1A1KDM4EKEAP1ARL3MBTL1
SCHEMBL31316614 0.80 MC4R (0.42) ALDH1A1KDM4EMAPTHRH3
SCHEMBL2783770 0.80 GAA (0.44) ALDH1A1KDM4EMAPTHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538091-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF Navitor Pharmaceuticals, Inc. (US) 2019-09-18 EP disclosed
WO-2018089499-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed