SCHEMBL20142746

SCHEMBL20142746

Cc1c(C#N)cccc1-n1ccnn1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 8/20 0.41
NISCH Q9Y2I1 1/20 0.38
KDM4E B2RXH2 1/20 0.38
KEAP1 Q14145 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
MAPT P10636 1/20 0.36
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
SLC6A9 P48067 1/20 0.36
TSHR P16473 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1587098 0.83 NOTUM (0.42) NOTUMKDM4EKEAP1SMN1; SMN2HIF1A
SCHEMBL30633068 0.83 NOTUM (0.42) NOTUMKDM4EKEAP1SMN1; SMN2HIF1A
SCHEMBL1587097 0.83 NOTUM (0.39) NOTUMKDM4EKEAP1SMN1; SMN2HIF1A
SCHEMBL18284703 0.81 NOTUM (0.38) NOTUMKDM4EKEAP1SMN1; SMN2HIF1A
SCHEMBL4531873 0.81 HCRTR1 (0.38) NOTUMKDM4EKEAP1HCRTR1HCRTR2
SCHEMBL2170102 0.79 NPC1 (0.46) NOTUMNISCHKDM4ESMN1; SMN2HIF1A
SCHEMBL18378736 0.78 NOTUM (0.47) NOTUMKEAP1SMN1; SMN2TSHRCYP1A2
SCHEMBL1586174 0.78 TSHR (0.43) NOTUMNISCHKDM4EKEAP1HCRTR1
SCHEMBL22702085 0.76 NOTUM (0.47) NOTUMKEAP1HCRTR1HCRTR2CYP1A2
SCHEMBL7111602 0.76 NOTUM (0.44) NOTUMKEAP1HCRTR1HCRTR2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021137665-A1 1, 2, 3-TRIAZOLE DERIVATIVE COMPOUND AS HSP90 INHIBITOR, AND USE THEREOF 이화여자대학교 산학협력단 2021-07-08 WO disclosed
EP-3538088-A1 HETEROCYCLIC MODULATORS OF LIPID SYNTHESIS 3-V Biosciences, Inc. (US) 2019-09-18 EP disclosed
US-9981942-B2 Piperidine derivatives having multimodal activity against pain LABORATORIOS DEL DR. ESTEVE S.A. (ES) 2018-05-29 US disclosed
WO-2018089904-A1 HETEROCYCLIC MODULATORS OF LIPID SYNTHESIS 3-V BIOSCIENCES, INC. (US) 2018-05-17 WO disclosed