SCHEMBL20142809

SCHEMBL20142809

CC1C(C(=O)NC(CC(=O)O)c2cc(Cl)cc(Cl)c2)CC12CN(C(=O)CCc1ccc3c(n1)NCCC3)C2

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 20/20 0.60
ITGAV P06756 20/20 0.60
ITGB5 P18084 13/20 0.60
ITGB6 P18564 11/20 0.60
ITGB8 P26012 10/20 0.60
ITGA2B P08514 5/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142676 0.87 ITGB3 (0.64) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20142679 0.87 ITGB3 (0.64) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20158347 0.85 ITGAV (0.76) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL30487498 0.81 ITGAV (0.54) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20158348 0.79 ITGAV (0.65) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20140735 0.79 ITGB3 (0.63) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20140736 0.79 ITGB3 (0.63) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20142297 0.78 ITGB3 (0.66) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20142900 0.78 ITGB3 (0.66) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20142299 0.78 ITGB3 (0.66) ITGB3ITGAVITGB5ITGB6ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538526-A1 CYCLOBUTANE- AND AZETIDINE-CONTAINING MONO AND SPIROCYCLIC COMPOUNDS AS ALPHA V INTEGRIN INHIBITORS Bristol-Myers Squibb Company (US) 2019-09-18 EP disclosed
WO-2018089355-A1 CYCLOBUTANE- AND AZETIDINE-CONTAINING MONO AND SPIROCYCLIC COMPOUNDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed