SCHEMBL20143997

SCHEMBL20143997

CC(C)c1cnc(NCc2cccc(F)n2)nc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.45
GRIN1 Q05586 4/20 0.42
GRIN2B Q13224 4/20 0.42
RXRA P19793 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
HDAC6 Q9UBN7 3/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC4 P56524 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
PDE1A P54750 2/20 0.37
PDE1B Q01064 2/20 0.37
PDE1C Q14123 2/20 0.37
CXCR4 P61073 1/20 0.36
ADORA2B P29275 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
VNN1 O95497 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15865881 0.83 ALOX5AP (0.50) ALOX5APGRIN1GRIN2BRXRAHDAC6
SCHEMBL13559933 0.81 CXCR4 (0.50) ALOX5APGRIN1GRIN2BRXRARAB9A
SCHEMBL13559731 0.79 ALOX5AP (0.50) ALOX5APGRIN1GRIN2BRXRANPC1
SCHEMBL8224027 0.77 HDAC3 (0.55) NPC1RAB9AHDAC6HDAC1MEN1
SCHEMBL13559904 0.76 ALOX5AP (0.47) ALOX5APGRIN1GRIN2BRXRANPC1
SCHEMBL19117565 0.71 NPC1 (0.61) NPC1RAB9AHDAC6HDAC1MEN1
SCHEMBL12536038 0.70 NPSR1 (0.41) ALOX5APCXCR4ADORA2BCYP3A4
SCHEMBL22804342 0.68 HDAC6 (0.78) HDAC6HDAC1HDAC4
SCHEMBL18503030 0.68 NPC1 (0.47) GRIN1GRIN2BRXRANPC1RAB9A
SCHEMBL26482966 0.67 RAB9A (0.44) GRIN1GRIN2BRXRANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2635566-B1 BENZIMIDAZOLE INHIBITORS OF LEUKOTRIENE PRODUCTION BOEHRINGER INGELHEIM INT (DE) 2018-05-16 EP disclosed