SCHEMBL20144912

SCHEMBL20144912

Cc1cnc(C(=O)N2CCCC(Nc3ccc(Cl)cn3)C2)c(-c2ncccn2)c1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 12/20 0.56
HCRTR2 O43614 5/20 0.53
CCNK O75909 3/20 0.47
CDK12 Q9NYV4 3/20 0.47
GFER P55789 1/20 0.46
CCNA2 P20248 1/20 0.44
CDK2 P24941 1/20 0.44
CDK7 P50613 1/20 0.44
CCNH P51946 1/20 0.44
MNAT1 P51948 1/20 0.44
GRM5 P41594 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20145115 0.93 HCRTR1 (0.56) HCRTR1HCRTR2CCNKCDK12GFER
SCHEMBL20144970 0.88 HCRTR1 (0.52) HCRTR1HCRTR2CCNKCDK12GFER
SCHEMBL20144789 0.87 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL18697684 0.87 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL20144927 0.86 HCRTR1 (0.70) HCRTR1HCRTR2CCNKCDK12GFER
SCHEMBL20145009 0.83 GFER (0.49) HCRTR1HCRTR2CCNKCDK12GFER
SCHEMBL20144876 0.81 HCRTR1 (0.69) HCRTR1HCRTR2
SCHEMBL16149117 0.81 HCRTR1 (0.77) HCRTR1HCRTR2
SCHEMBL20144983 0.79 HCRTR1 (0.52) HCRTR1HCRTR2CCNKCDK12
SCHEMBL20145164 0.79 HCRTR1 (0.52) HCRTR1HCRTR2CCNKCDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed