SCHEMBL20145009

SCHEMBL20145009

Cc1ccnc(C(=O)N2CCCC(Nc3ccc(Cl)cn3)C2)c1-c1ncccn1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GFER P55789 1/20 0.49
CCNK O75909 3/20 0.47
CDK12 Q9NYV4 3/20 0.47
HCRTR1 O43613 4/20 0.45
PROKR1 Q8TCW9 5/20 0.44
GRM5 P41594 2/20 0.44
KMT2A Q03164 1/20 0.43
HCRTR2 O43614 1/20 0.43
PLA2G1B P04054 1/20 0.43
ATG4B Q9Y4P1 1/20 0.43
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
CDK7 P50613 1/20 0.42
CCNH P51946 1/20 0.42
MNAT1 P51948 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20145008 0.87 HCRTR1 (0.53) HCRTR1PROKR1HCRTR2
SCHEMBL20144970 0.85 HCRTR1 (0.52) GFERCCNKCDK12HCRTR1GRM5
SCHEMBL20144912 0.83 HCRTR1 (0.56) GFERCCNKCDK12HCRTR1GRM5
SCHEMBL16148373 0.81 HCRTR1 (0.60) HCRTR1HCRTR2
SCHEMBL20145164 0.76 HCRTR1 (0.52) CCNKCDK12HCRTR1HCRTR2
SCHEMBL20144983 0.76 HCRTR1 (0.52) CCNKCDK12HCRTR1HCRTR2
SCHEMBL20144927 0.75 HCRTR1 (0.70) GFERCCNKCDK12HCRTR1PROKR1
SCHEMBL20145115 0.75 HCRTR1 (0.56) GFERCCNKCDK12HCRTR1KMT2A
SCHEMBL20145116 0.73 HCRTR1 (0.66) HCRTR1HCRTR2
SCHEMBL20144808 0.73 HCRTR1 (0.66) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed