SCHEMBL20145018

SCHEMBL20145018

Cc1ccc(C(=O)N2CCCC(Nc3ccc(C(F)(F)F)cn3)C2)c(N(N)/C=C\N)n1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 13/20 0.46
HCRTR2 O43614 11/20 0.44
MAP3K12 Q12852 1/20 0.43
PHGDH O43175 1/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
BLM P54132 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
HSD11B1 P28845 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20145082 0.91 HCRTR1 (0.45) HCRTR1HCRTR2PHGDHKMT2AMEN1
SCHEMBL20145022 0.90 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL18697657 0.80 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL20145007 0.80 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL18697767 0.77 HCRTR1 (0.72) HCRTR1HCRTR2
SCHEMBL20144987 0.77 HCRTR1 (0.72) HCRTR1HCRTR2
SCHEMBL20144729 0.77 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL20145031 0.75 HCRTR2 (0.70) HCRTR1HCRTR2
SCHEMBL20145056 0.75 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL20144723 0.75 HCRTR1 (0.70) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed