SCHEMBL20145082

SCHEMBL20145082

Cc1ccc(C(=O)N2CCCC(Nc3ncc(C(F)(F)F)cn3)C2)c(N(N)/C=C\N)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 8/20 0.45
HCRTR2 O43614 4/20 0.45
CCNK O75909 5/20 0.43
CDK12 Q9NYV4 5/20 0.43
MAPK3 P27361 2/20 0.39
GFER P55789 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39
BLM P54132 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
PHGDH O43175 1/20 0.38
CCNA2 P20248 2/20 0.38
CDK2 P24941 2/20 0.38
CDK7 P50613 2/20 0.38
CCNH P51946 2/20 0.38
MNAT1 P51948 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20145018 0.91 HCRTR1 (0.46) HCRTR1HCRTR2MEN1ALDH1A1POLB
SCHEMBL20145022 0.86 HCRTR1 (0.47) HCRTR1HCRTR2CCNKCDK12GFER
SCHEMBL20144867 0.79 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL20144729 0.77 HCRTR1 (0.46) HCRTR1HCRTR2GFER
SCHEMBL20145032 0.77 HCRTR1 (0.71) HCRTR1HCRTR2CCNKCDK12
SCHEMBL20144974 0.74 HCRTR1 (0.70) HCRTR1HCRTR2CCNKCDK12KMT2A
SCHEMBL20144821 0.74 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL20145111 0.73 CDK12 (0.46) HCRTR1HCRTR2CCNKCDK12MAPK3
SCHEMBL25226590 0.73 MAPK3 (0.50) HCRTR1HCRTR2CCNKCDK12MAPK3
SCHEMBL20144982 0.73 HCRTR1 (0.70) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed