SCHEMBL20145168

SCHEMBL20145168

O=C(c1ccccc1-c1ncccn1)N1CCC[C@@H](Oc2ncc(C(F)(F)F)cc2Cl)C1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 19/20 0.57
HCRTR2 O43614 7/20 0.51
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20145013 1.00 HCRTR1 (0.57) HCRTR1HCRTR2GAAMAPTCYP2C9
SCHEMBL18697567 0.93 HCRTR1 (0.58) HCRTR1HCRTR2
SCHEMBL20145077 0.93 HCRTR1 (0.58) HCRTR1HCRTR2
SCHEMBL20144914 0.91 HCRTR1 (0.69) HCRTR1HCRTR2
SCHEMBL20145027 0.91 HCRTR1 (0.59) HCRTR1HCRTR2
SCHEMBL18697758 0.91 HCRTR1 (0.69) HCRTR1HCRTR2
SCHEMBL20145015 0.90 HCRTR1 (0.51) HCRTR1HCRTR2GAAMAPTCYP2C9
SCHEMBL18697566 0.90 HCRTR1 (0.51) HCRTR1HCRTR2GAAMAPTCYP2C9
SCHEMBL20145090 0.87 HCRTR1 (0.59) HCRTR1HCRTR2
SCHEMBL20144872 0.86 HCRTR1 (0.67) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed