SCHEMBL2014553

SCHEMBL2014553

Cc1ccc(-n2nccn2)c(C(=O)N(C)C(CCNC(=O)c2cccn2C)Cc2ccccc2)c1

nearest known ligand 0.76

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 13/20 0.76
HCRTR2 O43614 12/20 0.76
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
PADI4 Q9UM07 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2015066 0.85 HCRTR1 (0.61) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2014992 0.83 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2051297 0.83 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2010789 0.82 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2015191 0.81 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL13139093 0.81 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL13139102 0.81 HCRTR1 (0.71) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2012749 0.80 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL13139060 0.80 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2011910 0.80 HCRTR1 (0.69) HCRTR1HCRTR2NPC1RAB9APADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed