SCHEMBL20145802

SCHEMBL20145802

CN(C)C(=O)C1CCN(c2ncnc(N)c2F)CC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP46A1 Q9Y6A2 8/20 0.47
NEK2 P51955 1/20 0.43
PIK3CD O00329 1/20 0.41
ATR Q13535 2/20 0.41
PDE10A Q9Y233 1/20 0.40
AKT2 P31751 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
RPS6KB1 P23443 2/20 0.38
SYK P43405 1/20 0.38
BTK Q06187 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20145794 0.84 AKT2 (0.55) NEK2AKT2ALDH1A1HSD17B10
SCHEMBL20145894 0.82 MAP4K4 (0.52) CYP46A1NEK2ATRPDE10AAKT2
SCHEMBL22240433 0.79 UBE2N (0.54) ATR
SCHEMBL19801719 0.74 RPS6KB1 (0.42) AKT2RPS6KB1BTK
SCHEMBL14334180 0.73 MALT1 (0.52) CYP46A1NEK2PDE10AALDH1A1
SCHEMBL22240510 0.72 BTK (0.47) NEK2BTK
SCHEMBL25668037 0.72 NEK2 (0.49) NEK2BTK
SCHEMBL16786557 0.72 BTK (0.41) BTK
SCHEMBL16786552 0.72 BTK (0.41) BTK
SCHEMBL20862434 0.72 MAP4K4 (0.48) PIK3CDRPS6KB1BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2858499-B1 PYRIMIDINYL TYROSINE KINASE INHIBITORS BIOGEN MA INC (US) 2018-05-16 EP disclosed