SCHEMBL2014739

SCHEMBL2014739

CCCCOC(=O)NC(CCC(=O)O)C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 8/20 0.45
CTSS P25774 3/20 0.45
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
PLA2G2C Q5R387 1/20 0.39
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
FOLH1 Q04609 5/20 0.37
NOD1 Q9Y239 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4365404 1.00 CTSK (0.45) CTSKCTSSBCHEACHEPLA2G2C
SCHEMBL15457738 0.89 CTSK (0.51) CTSKCTSSBCHEACHECYP1A2
SCHEMBL13983158 0.89 CTSK (0.51) CTSKCTSSBCHEACHECYP1A2
SCHEMBL28190852 0.89 CTSK (0.55) CTSKCTSS
SCHEMBL5623720 0.86 CTSK (0.44) CTSKCTSSACHE
SCHEMBL4362188 0.86 CTSK (0.44) CTSKCTSSACHE
SCHEMBL7284821 0.85 BCHE (0.52) CTSKCTSSBCHEACHEPLA2G2C
SCHEMBL7288988 0.85 BCHE (0.52) CTSKCTSSBCHEACHEPLA2G2C
SCHEMBL19692119 0.85 CTSK (0.45) CTSKCTSSACHECYP1A2CYP2C9
SCHEMBL7006306 0.85 KMT2A (0.49) PLA2G2CITGB3ITGA2BFOLH1NOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3197885-A2 HETEROCYCLIC COMPOUNDS AND USE THEREOF Chao, Yu-Sheng (US) 2017-08-02 EP disclosed
WO-2016048861-A2 HETEROCYCLIC COMPOUNDS AND USE THEREOF NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2016-03-31 WO disclosed
WO-2011067266-A1 CARBOXYLIC ACID ANALOGS AS GLYCOGEN SYNTHASE ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-09 WO disclosed
EP-1230243-A1 POYCYLOALKYLPURINES AS ADENOSINE RECEPTOR ANTAGONISTS BIOGEN, INC. (US) 2002-08-14 EP disclosed
WO-2001034610-A1 POLYCYCLOALKYLPURINES AS ADENOSINE RECEPTOR ANTAGONISTS BIOGEN, INC. (US) 2001-05-17 WO disclosed