SCHEMBL2014753

SCHEMBL2014753

CN(C(=O)c1ccc2ncccc2c1)C(CCCNC(=O)c1cccn1C)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.46
HCRTR2 O43614 1/20 0.46
HTR1A P08908 1/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
ADRA1D P25100 1/20 0.46
HTR2A P28223 1/20 0.46
ADRA1A P35348 1/20 0.46
HRH1 P35367 1/20 0.46
ADRA1B P35368 1/20 0.46
DRD3 P35462 1/20 0.46
KCNH2 Q12809 1/20 0.46
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
PLK1 P53350 1/20 0.39
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014754 1.00 HCRTR1 (0.46) HCRTR1HCRTR2HTR1AADRA2AADRA2B
SCHEMBL2016049 0.90 HCRTR1 (0.46) HCRTR1HCRTR2HTR1AHTR2ADRD3
SCHEMBL2016048 0.90 HCRTR1 (0.46) HCRTR1HCRTR2HTR1AHTR2ADRD3
SCHEMBL2013785 0.84 HCRTR1 (0.67) HCRTR1HCRTR2HTR1AADRA2AADRA2B
SCHEMBL2011909 0.83 HCRTR1 (0.45) HCRTR1HCRTR2ADRA1DADRA1AADRA1B
SCHEMBL2011913 0.83 HCRTR1 (0.45) HCRTR1HCRTR2ADRA1DADRA1AADRA1B
SCHEMBL2050042 0.74 NPC1 (0.38) HCRTR1HCRTR2ADRA1DADRA1AADRA1B
SCHEMBL2013242 0.74 HCRTR1 (0.70) HCRTR1HCRTR2ALDH1A1NPC1RAB9A
SCHEMBL2015950 0.74 HCRTR1 (0.70) HCRTR1HCRTR2ALDH1A1NPC1RAB9A
SCHEMBL6918071 0.73 HCRTR1 (0.66) HCRTR1HCRTR2HTR1AHTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed