SCHEMBL20148914

SCHEMBL20148914

CNc1c(N)nc(-c2nn(Cc3ccccc3F)c3ncccc23)nc1N

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.67
KCNH2 Q12809 1/20 0.67
PDE5A O76074 12/20 0.56
GUCY1A1 Q02108 6/20 0.54
GUCY1B1 Q02153 6/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL255818 0.90 ADORA3 (0.65) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL15127590 0.89 ADORA3 (0.64) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL174210 0.89 ADORA3 (0.64) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL29154434 0.89 ADORA3 (0.68) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL174847 0.88 ADORA3 (0.67) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL23434879 0.88 ADORA3 (0.67) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL255851 0.88 ADORA3 (0.62) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL18212217 0.88 ADORA3 (0.70) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
Hydrochloric Acid SCHEMBL1930775 0.87 ADORA3 (0.66) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
Hydrochloric Acid SCHEMBL18496411 0.87 ADORA3 (0.66) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089328-A1 TREATMENT OF CNS DISEASES WITH SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
CN-105367568-A Riociguat preparation method ZHEJIANG JINGXIN PHARMACEUTICAL CO LTD 2016-03-02 CN disclosed
CN-105367568-A Riociguat preparation method ZHEJIANG JINGXIN PHARMACEUTICAL CO LTD 2016-03-02 CN disclosed
CN-105367567-A Compound and application thereof in preparation of riociguat ZHEJIANG JINGXIN PHARMACEUTICAL CO LTD 2016-03-02 CN disclosed
CN-105367567-A Compound and application thereof in preparation of riociguat ZHEJIANG JINGXIN PHARMACEUTICAL CO LTD 2016-03-02 CN disclosed