SCHEMBL2015135

SCHEMBL2015135

Cc1noc(C)c1C(=O)N(C)C(CCNC(=O)c1cccn1C)Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.59
HCRTR2 O43614 2/20 0.59
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
TSHR P16473 1/20 0.46
GAA P10253 1/20 0.44
TAS2R8 Q9NYW2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.38
PADI4 Q9UM07 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2054315 0.91 HCRTR1 (0.57) HCRTR1HCRTR2NPC1RAB9ATSHR
SCHEMBL2049937 0.91 HCRTR1 (0.57) HCRTR1HCRTR2NPC1RAB9ATSHR
SCHEMBL2015329 0.91 HCRTR1 (0.57) HCRTR1HCRTR2NPC1RAB9ATSHR
SCHEMBL2010469 0.91 HCRTR1 (0.57) HCRTR1HCRTR2NPC1RAB9ATSHR
SCHEMBL2054212 0.85 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2054210 0.85 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2010838 0.83 HCRTR1 (0.63) HCRTR1HCRTR2NPC1RAB9ATSHR
SCHEMBL2012339 0.83 HCRTR1 (0.63) HCRTR1HCRTR2NPC1RAB9ATAS2R8
SCHEMBL13139060 0.83 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2012675 0.83 HCRTR1 (0.57) HCRTR1HCRTR2NPC1RAB9APADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed