SCHEMBL2015329

SCHEMBL2015329

Cc1onc(-c2ccccc2)c1C(=O)N(C)C(CCNC(=O)c1cccn1C)Cc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.57
HCRTR2 O43614 2/20 0.57
L3MBTL1 Q9Y468 1/20 0.48
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 1/20 0.44
HDAC6 Q9UBN7 4/20 0.43
HDAC3 O15379 2/20 0.43
NCOR2 Q9Y618 2/20 0.43
ALDH1A1 P00352 3/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC4 P56524 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2049937 1.00 HCRTR1 (0.57) HCRTR1HCRTR2L3MBTL1NPC1RAB9A
SCHEMBL2015135 0.91 HCRTR1 (0.59) HCRTR1HCRTR2L3MBTL1NPC1RAB9A
SCHEMBL2010469 0.87 HCRTR1 (0.57) HCRTR1HCRTR2L3MBTL1NPC1RAB9A
SCHEMBL2054315 0.87 HCRTR1 (0.57) HCRTR1HCRTR2L3MBTL1NPC1RAB9A
SCHEMBL2054210 0.81 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9AKMT2A
SCHEMBL2054212 0.81 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9AKMT2A
SCHEMBL13139060 0.81 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9AKMT2A
SCHEMBL2010539 0.80 HCRTR1 (0.63) HCRTR1HCRTR2NPC1RAB9AHDAC6
SCHEMBL6919915 0.80 HCRTR1 (0.65) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL2015468 0.80 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed