SCHEMBL2015255

SCHEMBL2015255

OCCc1cc2ncccc2nc1-c1cccc(F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
PTGDR2 Q9Y5Y4 3/20 0.39
ADORA2A P29274 2/20 0.39
TBXA2R P21731 1/20 0.38
PTGDR Q13258 1/20 0.38
SYK P43405 1/20 0.38
PDE4A P27815 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36
CSNK2A2 P19784 1/20 0.36
CSNK2B P67870 1/20 0.36
CLK4 Q9HAZ1 2/20 0.36
CDC7 O00311 1/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36
PIM1 P11309 1/20 0.36
PRKACA P17612 1/20 0.36
CDK2 P24941 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1989452 0.90 BCHE (0.46) BCHEACHEPTGDR2ADORA2ATBXA2R
SCHEMBL2015151 0.87 SYK (0.45) BCHEACHEPTGDR2ADORA2ATBXA2R
SCHEMBL9952652 0.84 BCHE (0.46) BCHEACHEPTGDR2ADORA2ATBXA2R
SCHEMBL1988633 0.80 BCHE (0.44) BCHEACHEADORA2APDE4APDE4B
SCHEMBL4435275 0.79 NT5E (0.44) PTGDR2ADORA2ATBXA2RPTGDRCSNK2A2
SCHEMBL12629115 0.77 ADORA2A (0.50) BCHEACHEADORA2ASYKCLK4
SCHEMBL1989290 0.76 MAPK14 (0.38) BCHEACHESYKCYP1A2CYP3A4
SCHEMBL1990582 0.74 BCHE (0.44) BCHEACHEADORA2ASYKCLK4
SCHEMBL1991506 0.74 BCHE (0.46) BCHEACHEADORA2ACLK4CDC7
SCHEMBL1988818 0.74 BCHE (0.46) BCHEACHEADORA2ASYKPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513109-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES Amgen Inc. (US) 2012-10-24 EP disclosed
WO-2011075628-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2011-06-23 WO disclosed