SCHEMBL20153341

SCHEMBL20153341

CCOC(=O)CCn1ccc(CCCc2ccc3c(n2)NCCC3)n1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.47
ITGB3 P05106 17/20 0.47
ITGA2B P08514 4/20 0.47
ITGB6 P18564 9/20 0.45
ITGB5 P18084 5/20 0.45
ITGB8 P26012 5/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20153399 0.86 ITGB3 (0.59) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL6265738 0.85 ITGAV (0.56) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL19809630 0.84 ITGAV (0.61) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL22223353 0.83 ITGAV (0.60) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL16607379 0.83 ITGAV (0.60) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL5252354 0.83 ITGAV (0.53) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL29860519 0.82 ITGB3 (0.58) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL22223273 0.81 ITGAV (0.54) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL5247260 0.81 ITGAV (0.57) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL2491969 0.80 ITGAV (0.60) ITGAVITGB3ITGA2BITGB6ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538525-B1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-06-22 EP disclosed
WO-2018089353-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed